SCHEMBL14865359

SCHEMBL14865359

COc1ccc(C(=O)NC2(C(=O)NCc3ccc(Nc4ccc(Br)cc4C(F)(F)I)cn3)CC2)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 2/20 0.35
BDKRB1 P46663 2/20 0.34
EPHX2 P34913 1/20 0.34
GPR183 P32249 1/20 0.34
KCNH2 Q12809 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN9A Q15858 1/20 0.33
GPR35 Q9HC97 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
HDAC1 Q13547 2/20 0.33
PIK3CA P42336 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
USP2 O75604 1/20 0.33
PABPC1 P11940 1/20 0.33
MAPK1 P28482 1/20 0.33
CXCR1 P25024 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186380 0.94 BDKRB1 (0.37) MEN1KMT2AMAPTBDKRB1EPHX2
SCHEMBL186047 0.85 MEN1 (0.43) MEN1KMT2AMAPTBDKRB1EPHX2
SCHEMBL2805112 0.85 BDKRB1 (0.37) BDKRB1KCNH2SCN5ASCN9AHDAC1
SCHEMBL185963 0.84 FPR2 (0.39) MEN1KMT2ABDKRB1HDAC1CTSL
SCHEMBL185691 0.84 CNR2 (0.38) BDKRB1CTSLCTSBCTSS
SCHEMBL186154 0.83 CNR2 (0.37) BDKRB1EPHX2HDAC1CTSLCTSB
SCHEMBL186861 0.83 CNR2 (0.37) BDKRB1EPHX2CTSLCTSBCTSS
SCHEMBL13128577 0.83 CNR2 (0.36) MAPTBDKRB1EPHX2HDAC1CTSL
SCHEMBL2805326 0.83 CNR2 (0.37) BDKRB1SCN9AHDAC1CTSLCTSB
SCHEMBL186671 0.82 CNR2 (0.37) BDKRB1CTSLCTSBCTSSCXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed