SCHEMBL14865408

SCHEMBL14865408

O=C(NCc1ncc(Nc2ccccc2C(F)(F)F)cc1Cl)[C@@H]1CCOC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.39
EPHX2 P34913 3/20 0.39
P2RX7 Q99572 6/20 0.39
MAPK10 P53779 3/20 0.38
PIP5K1C O60331 2/20 0.38
PIK3CA P42336 2/20 0.38
MAPK8 P45983 2/20 0.38
MAPK14 Q16539 2/20 0.38
PIP5K1B O14986 1/20 0.38
PIP5K1A Q99755 1/20 0.38
CNR2 P34972 5/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13160089 0.90 MAPK10 (0.42) EPHX2P2RX7MAPK10PIP5K1CPIK3CA
SCHEMBL13160304 0.90 EPHX2 (0.40) CYP2C9EPHX2MAPK10PIP5K1CPIK3CA
SCHEMBL13160246 0.87 HTR1A (0.40) CYP2C9EPHX2P2RX7MAPK10PIP5K1C
SCHEMBL13160140 0.83 CNR2 (0.42) CYP2C9EPHX2MAPK10MAPK8MAPK14
SCHEMBL13159674 0.81 MAPK10 (0.44) EPHX2P2RX7MAPK10PIP5K1CPIK3CA
SCHEMBL185656 0.81 DHODH (0.40) CNR2
SCHEMBL13159831 0.80 EPHX2 (0.42) CYP2C9EPHX2MAPK10PIP5K1CPIK3CA
SCHEMBL13159669 0.80 EPHX2 (0.42) CYP2C9EPHX2MAPK10PIP5K1CPIK3CA
SCHEMBL13159680 0.80 MAPK10 (0.42) EPHX2P2RX7MAPK10PIP5K1CPIK3CA
SCHEMBL14865420 0.79 HTR1A (0.41) CYP2C9EPHX2P2RX7MAPK10PIP5K1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed