SCHEMBL14869717

SCHEMBL14869717

NC(=O)c1ccccc1C1CCNC1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.54
JAK3 P52333 1/20 0.48
IKBKB O14920 2/20 0.47
CHUK O15111 2/20 0.47
CSF1R P07333 1/20 0.47
BTK Q06187 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.45
CYP2D6 P10635 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KCNH2 Q12809 1/20 0.44
ADRA1A P35348 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5968190 1.00 PARP1 (0.54) PARP1JAK3IKBKBCHUKCSF1R
SCHEMBL5330092 1.00 PARP1 (0.54) PARP1JAK3IKBKBCHUKCSF1R
Hydrochloric Acid SCHEMBL28155977 0.98 PARP1 (0.53) PARP1JAK3IKBKBCHUKCSF1R
Hydrochloric Acid SCHEMBL3669412 0.98 PARP1 (0.53) PARP1JAK3IKBKBCHUKCSF1R
Hydrochloric Acid SCHEMBL28155968 0.98 PARP1 (0.53) PARP1JAK3IKBKBCHUKCSF1R
SCHEMBL31227227 0.91 CSF1R (0.57) PARP1IKBKBCHUKCSF1RBTK
SCHEMBL31227274 0.91 CSF1R (0.57) PARP1IKBKBCHUKCSF1RBTK
SCHEMBL3649878 0.91 CSF1R (0.57) PARP1IKBKBCHUKCSF1RBTK
SCHEMBL1006493 0.90 IKBKB (0.53) PARP1IKBKBCHUKSIRT2SLC6A2
Hydrochloric Acid SCHEMBL16445630 0.89 CSF1R (0.56) PARP1IKBKBCHUKCSF1RBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021239117-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI) , INC. (CN) 2021-12-02 WO disclosed
US-9067930-B2 2-oxo-piperidinyl derivatives UCB PHARMA, S.A. (BE) 2015-06-30 US disclosed
US-9067930-B2 2-oxo-piperidinyl derivatives UCB PHARMA, S.A. (BE) 2015-06-30 US disclosed
US-9067930-B2 2-oxo-piperidinyl derivatives UCB PHARMA, S.A. (BE) 2015-06-30 US disclosed
EP-2766353-B1 2-OXO-PIPERIDINYL DERIVATIVES UCB PHARMA SA (BE) 2015-06-17 EP disclosed
US-20150011526-A1 2-Oxo-Piperidinyl Derivatives UCB BIOPHARMA SPRL (BE) 2015-01-08 US disclosed
US-20150011526-A1 2-Oxo-Piperidinyl Derivatives UCB BIOPHARMA SPRL (BE) 2015-01-08 US disclosed
US-20150011526-A1 2-Oxo-Piperidinyl Derivatives UCB BIOPHARMA SPRL (BE) 2015-01-08 US disclosed
EP-2766353-A1 2-OXO-PIPERIDINYL DERIVATIVES UCB Pharma, S.A. (BE) 2014-08-20 EP disclosed
WO-2013053725-A1 2-OXO-PIPERIDINYL DERIVATIVES UCB PHARMA, S.A. (BE) 2013-04-18 WO disclosed
WO-2013053725-A1 2-OXO-PIPERIDINYL DERIVATIVES UCB PHARMA, S.A. (BE) 2013-04-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150011526-A1 2-Oxo-Piperidinyl Derivatives CYP3A4, CYP2C19, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 PARP1 400/4885JAK3 2001/4885IKBKB 1899/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.