SCHEMBL14879201

SCHEMBL14879201

COC(=O)N[C@@H](Cc1cscn1)C(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.44
CTSK P43235 2/20 0.42
CAPN1 P07384 1/20 0.41
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
HDAC6 Q9UBN7 6/20 0.39
HDAC1 Q13547 4/20 0.39
SCN9A Q15858 1/20 0.39
FOLH1 Q04609 1/20 0.38
GPR142 Q7Z601 1/20 0.38
DPP4 P27487 2/20 0.36
DPP8 Q6V1X1 2/20 0.36
DPP9 Q86TI2 2/20 0.36
NLRP3 Q96P20 1/20 0.35
ATM Q13315 1/20 0.35
LCK P06239 1/20 0.35
KLKB1 P03952 1/20 0.35
ALDH1A1 P00352 1/20 0.35
THRB P10828 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL756368 0.89 FOLH1 (0.47) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL18731295 0.89 FOLH1 (0.47) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL14864797 0.89 CTSK (0.42) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL23324594 0.88 SCN9A (0.50) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL25888951 0.88 SCN9A (0.50) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL888810 0.86 CTSK (0.43) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL10122815 0.86 CTSK (0.43) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL14886205 0.86 CTSK (0.43) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL12762220 0.85 CNR2 (0.41) CNR2CTSKCAPN1CTSBCTSS
SCHEMBL16574843 0.85 CNR2 (0.41) CNR2CTSKCAPN1CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242750-B1 CONFORMATIONALLY RESTRICTED BIPHENYL DERIVATIVES FOR USE AS HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2013-04-24 EP disclosed