SCHEMBL1488705

SCHEMBL1488705

C=Cc1c(C)cc(-c2nnc(N(CC3CC3)C(=O)Cc3ccccc3Cl)s2)cc1C

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 13/20 0.47
KDM4E B2RXH2 3/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
GAA P10253 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
CPB1 P15086 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
S1PR3 Q99500 2/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TAS2R14 Q9NYV8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489004 0.81 S1PR1 (0.56) S1PR1S1PR3
SCHEMBL1488957 0.80 S1PR1 (0.51) S1PR1KDM4EMEN1CYP1A2GAA
SCHEMBL1489747 0.76 S1PR1 (0.49) S1PR1KDM4EALDH1A1HSD17B10TP53
SCHEMBL1489950 0.75 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL2300588 0.73 S1PR1 (0.49) S1PR1KDM4EMEN1CYP1A2GAA
SCHEMBL1489469 0.73 S1PR1 (0.50) S1PR1KDM4EALDH1A1HSD17B10TP53
SCHEMBL2300611 0.72 S1PR1 (0.57) S1PR1S1PR3
SCHEMBL1489180 0.72 S1PR1 (0.69) S1PR1CPB1S1PR3
SCHEMBL2297250 0.71 S1PR1 (0.53) S1PR1KDM4EALDH1A1HSD17B10TP53
SCHEMBL1489133 0.70 S1PR1 (0.47) S1PR1KDM4EGAAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed