SCHEMBL14896356

SCHEMBL14896356

N#Cc1cccc(C2OCCCO2)c1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
LRRK2 Q5S007 7/20 0.34
EGFR P00533 1/20 0.34
BCAT1 P54687 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
USP30 Q70CQ3 1/20 0.32
OPRL1 P41146 1/20 0.32
KMT2A Q03164 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20592264 0.77 TSHR (0.39) CYP11B1CYP11B2SLC6A2SLC6A4SLC6A3
SCHEMBL29209742 0.75 OPRL1 (0.39) SLC6A2SLC6A4SLC6A3HTR2CHTR2B
SCHEMBL30881887 0.75 OPRL1 (0.39) SLC6A2SLC6A4SLC6A3HTR2CHTR2B
SCHEMBL14896357 0.75 MAPKAPK2 (0.35) CYP11B1CYP11B2SLC6A2SLC6A4SLC6A3
SCHEMBL28604214 0.75 PDCD1 (0.42) HTR2CHTR2BKDM4EALDH1A1OPRL1
SCHEMBL28771523 0.73 PRKACA (0.49) HTR2CHTR2B
SCHEMBL122002 0.72 CYP11B2 (0.43) CYP11B1CYP11B2AR
SCHEMBL24416920 0.71 CYP11B1 (0.42) CYP11B1CYP11B2SLC6A4HTR2CHTR2B
SCHEMBL21873113 0.71 KDM4E (0.40) CYP11B1CYP11B2KDM4EALDH1A1
SCHEMBL29713462 0.71 KDM4E (0.40) CYP11B1CYP11B2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013062837-A1 PIPERIDINE DERIVATIVES USEFUL AS GPR119 AGONISTS MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed