SCHEMBL14899016

SCHEMBL14899016

C=C(C)C1(C(NC(=O)OC(C)(C)C)C(=O)O)CCC1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
CTSL P07711 3/20 0.34
CTSK P43235 11/20 0.33
CTSS P25774 7/20 0.33
CTSB P07858 2/20 0.32
BTK Q06187 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14216682 0.97 CA1 (0.35) CA1CA2CA7KMT2AMEN1
SCHEMBL14899013 0.87 CA1 (0.34) CA1CA2CA7KMT2AMEN1
SCHEMBL12936848 0.84 CA1 (0.34) CA1CA2CA7KMT2AMEN1
SCHEMBL9509419 0.82 CA1 (0.40) CA1CA2CA7KMT2AMEN1
SCHEMBL15105800 0.80 CA1 (0.39) CA1CA2CA7KMT2AMEN1
SCHEMBL28269476 0.80 CA1 (0.39) CA1CA2CA7KMT2AMEN1
SCHEMBL9825794 0.79 CA1 (0.38) CA1CA2CA7KMT2AMEN1
SCHEMBL15105955 0.79 CA1 (0.40) CA1CA2CA7KMT2AMEN1
SCHEMBL2377942 0.79 CA1 (0.40) CA1CA2CA7KMT2AMEN1
SCHEMBL2377936 0.79 CA1 (0.40) CA1CA2CA7KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44186-E1 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-30 US disclosed
US-RE44186-E1 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-30 US disclosed