SCHEMBL14899720

SCHEMBL14899720

COSCc1ccc(I)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 11/20 0.52
CYP3A4 P08684 3/20 0.41
IDO1 P14902 2/20 0.41
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2E1 P05181 1/20 0.38
CYP2C8 P10632 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
DAO P14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8824002 0.81 APP (0.46) APPCYP3A4IDO1DAO
SCHEMBL3353930 0.79 IDO1 (0.47) IDO1CYP1A2
SCHEMBL14899725 0.77 TDP1 (0.44) CYP3A4IDO1
SCHEMBL546541 0.76 CYP1A2 (0.42) CYP3A4IDO1CYP1A2CYP2D6CYP2C19
SCHEMBL514628 0.73 APP (0.47) APPCYP3A4IDO1CYP1A2CYP2D6
SCHEMBL8824005 0.72 APP (0.45) APPCYP3A4IDO1CYP1A2CYP2D6
Methylene Chloride SCHEMBL28192144 0.71 CYP1A2 (0.38) CYP3A4IDO1CYP1A2CYP2D6
SCHEMBL13271320 0.70 APP (0.44) APPCYP3A4IDO1CYP1A2CYP2D6
SCHEMBL8007514 0.70 APP (0.44) APPCYP3A4IDO1CYP1A2CYP2D6
SCHEMBL18475586 0.69 APP (1.00) APPCYP3A4IDO1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2586778-A2 Pyridazinone derivatives useful as glucan synthase inhibitors Merck Sharp & Dohme Corp. (US) 2013-05-01 EP disclosed