SCHEMBL14906387

SCHEMBL14906387

Fc1ccc(Cl)c(-c2ccncc2-n2cncc2-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 16/20 0.40
PDE2A O00408 1/20 0.35
PDE10A Q9Y233 1/20 0.35
KCNA5 P22460 1/20 0.33
KCNH2 Q12809 1/20 0.33
RPS6KA3 P51812 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14906407 0.91 GPBAR1 (0.40) GPBAR1PDE2APDE10A
SCHEMBL14906389 0.87 GPBAR1 (0.47) GPBAR1
SCHEMBL14906396 0.87 GPBAR1 (0.47) GPBAR1
SCHEMBL14906364 0.86 GPBAR1 (0.37) GPBAR1
SCHEMBL14906381 0.85 SRC (0.38) GPBAR1RPS6KA3
SCHEMBL14906383 0.85 GPBAR1 (0.49) GPBAR1
SCHEMBL14906367 0.85 KLRK1 (0.39) GPBAR1PDE2APDE10A
SCHEMBL14906413 0.85 GPBAR1 (0.39) GPBAR1PDE2APDE10A
SCHEMBL14906380 0.83 GPBAR1 (0.42) GPBAR1KCNA5KCNH2
SCHEMBL14906397 0.83 GPBAR1 (0.39) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013062887-A1 SUBSTITUTED PYRIDINE DERIVATIVES USEFUL AS GPR131 AGONISTS MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed