SCHEMBL14906381

SCHEMBL14906381

Fc1ccc(-c2ccncc2-n2cncc2-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.38
BRAF P15056 1/20 0.38
KDR P35968 1/20 0.38
RPS6KA3 P51812 2/20 0.38
GPBAR1 Q8TDU6 8/20 0.37
KLRK1 P26718 2/20 0.35
MICA Q29983 2/20 0.35
RAET1L Q5VY80 2/20 0.35
HSP90AA1 P07900 2/20 0.35
HSP90AB1 P08238 2/20 0.35
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CYP1A2 P05177 1/20 0.34
METAP2 P50579 1/20 0.34
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14906370 0.89 GPBAR1 (0.40) GPBAR1KLRK1MICARAET1LHSP90AA1
SCHEMBL14906516 0.89 GPBAR1 (0.47) GPBAR1METAP2
SCHEMBL14906389 0.87 GPBAR1 (0.47) GPBAR1CYP1A2METAP2
SCHEMBL14906364 0.86 GPBAR1 (0.37) GPBAR1S1PR1S1PR3GSK3AGSK3B
SCHEMBL14906387 0.85 GPBAR1 (0.40) RPS6KA3GPBAR1
SCHEMBL14906383 0.85 GPBAR1 (0.49) GPBAR1CYP1A2METAP2
SCHEMBL14906367 0.85 KLRK1 (0.39) GPBAR1KLRK1MICARAET1LS1PR1
SCHEMBL14906417 0.85 GPBAR1 (0.36) GPBAR1KLRK1MICARAET1LHSP90AA1
SCHEMBL14896119 0.83 GPBAR1 (0.52) GPBAR1
SCHEMBL14906369 0.83 IDO1 (0.42) KDRGPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013062887-A1 SUBSTITUTED PYRIDINE DERIVATIVES USEFUL AS GPR131 AGONISTS MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed