SCHEMBL14907679

SCHEMBL14907679

NCCCC(=O)NCc1ccnc2[nH]ccc12

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
AKT1 P31749 2/20 0.41
NUDT1 P36639 2/20 0.40
IKBKB O14920 2/20 0.40
CHUK O15111 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
RET P07949 1/20 0.39
NEK1 Q96PY6 1/20 0.39
KLKB1 P03952 1/20 0.38
CIT O14578 3/20 0.38
TPSAB1 Q15661 1/20 0.38
PRKCI P41743 3/20 0.38
ROCK1 Q13464 1/20 0.38
AXL P30530 1/20 0.38
MAPT P10636 1/20 0.37
JAK2 O60674 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14907682 0.84 AKT1 (0.43) AKT1NUDT1IKBKBCHUKRET
SCHEMBL14907656 0.81 AKT1 (0.49) AKT1NUDT1IKBKBCHUKNEK1
SCHEMBL14907651 0.79 AKT1 (0.38) AKT1NUDT1IKBKBCHUKRET
SCHEMBL14907989 0.78 AKT1 (0.38) AKT1NUDT1IKBKBCHUKRET
SCHEMBL14907655 0.77 RET (0.43) CYP3A4NUDT1RETCITPRKCI
SCHEMBL14907690 0.77 RET (0.37) NUDT1IKBKBCHUKRETNEK1
SCHEMBL14907678 0.76 HTT (0.52) RETROCK1JAK2HDAC6
SCHEMBL14907662 0.76 NUDT1 (0.44) AKT1NUDT1IKBKBCHUKRET
SCHEMBL14907834 0.76 JAK2 (0.41) AKT1NUDT1IKBKBCHUKRET
SCHEMBL14907663 0.75 AKT1 (0.44) AKT1NUDT1IKBKBCHUKRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9174984-B2 Chemical compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2015-11-03 US disclosed
US-20140296204-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2014-10-02 US disclosed
WO-2013062945-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2013-05-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296204-A1 CHEMICAL COMPOUNDS DNMT1, DNMT3A, DNMT3B CYP3A4 438/4885AKT1 887/4885NUDT1 829/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.