SCHEMBL14909074

SCHEMBL14909074

CC(C)(C)N(C[C@H](Nc1nc(Cl)c(C#N)cc1F)C1CC1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.34
ACHE P22303 4/20 0.33
BCHE P06276 3/20 0.33
JAK2 O60674 1/20 0.31
JAK3 P52333 1/20 0.31
SOS1 Q07889 2/20 0.31
S1PR3 Q99500 1/20 0.31
PGR P06401 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14909075 1.00 KHK (0.34) KHKACHEBCHEJAK2JAK3
SCHEMBL14910361 0.85 KHK (0.37) KHKACHEBCHES1PR3
SCHEMBL14910363 0.85 KHK (0.37) KHKACHEBCHES1PR3
SCHEMBL14909736 0.85 ACHE (0.34) KHKACHEBCHEJAK2JAK3
SCHEMBL14909735 0.85 ACHE (0.34) KHKACHEBCHEJAK2JAK3
SCHEMBL14911191 0.83 KHK (0.36) KHK
SCHEMBL14911192 0.83 KHK (0.36) KHK
SCHEMBL14909516 0.82 KHK (0.34) KHK
SCHEMBL14908685 0.82 KHK (0.34) KHK
SCHEMBL14911504 0.82 KHK (0.34) KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2589592-B1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM CORP (JP) 2018-08-22 EP disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed