SCHEMBL14910883

SCHEMBL14910883

Cc1cc(OC(F)F)ccc1-c1cc(N)[nH]n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 3/20 0.39
CA9 Q16790 1/20 0.39
KCNH2 Q12809 2/20 0.38
DRD1 P21728 2/20 0.38
CYP1A2 P05177 2/20 0.36
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
LMNA P02545 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
CRHR1 P34998 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853118 0.78 MAPT (0.41) ALPLCA9DRD1CYP1A2GAA
SCHEMBL14910385 0.76 TLR8 (0.42) ALPLCA9GAAKDM4ENPC1
SCHEMBL4856665 0.76 ALPL (0.58) ALPLCA9GAAKDM4ENPC1
SCHEMBL2088520 0.74 MAP4K4 (0.50) KCNH2DRD1GAAADORA1
SCHEMBL2091970 0.74 PARP15 (0.39) KCNH2ADORA2APPARG
SCHEMBL5305952 0.73 NPC1 (0.41) ALPLCA9GAAKDM4ENPC1
SCHEMBL14726304 0.73 NOTUM (0.48) ALPLCA9GAAKDM4ENPC1
SCHEMBL1857325 0.72 DRD1 (0.40) DRD1CYP1A2GAAKDM4ENPC1
SCHEMBL14910882 0.71 APP (0.31)
SCHEMBL1857868 0.71 NPC1 (0.54) CYP1A2GAAKDM4ENPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118067-B1 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS SIENA BIOTECH SPA (IT) 2013-05-08 EP disclosed