SCHEMBL14918170

SCHEMBL14918170

FC(F)(F)c1nc(-c2cnc(CNc3ccnc(-c4cccnc4)n3)nc2)no1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 14/20 0.63
HDAC1 Q13547 12/20 0.63
HDAC4 P56524 8/20 0.63
HDAC8 Q9BY41 6/20 0.56
CLK4 Q9HAZ1 6/20 0.55
CYP1A2 P05177 4/20 0.55
CYP3A4 P08684 4/20 0.55
CYP2D6 P10635 4/20 0.55
CYP2C19 P33261 3/20 0.55
ALOX15 P16050 2/20 0.55
USP2 O75604 1/20 0.54
CYP2C9 P11712 2/20 0.53
MAPK1 P28482 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HSD17B10 Q99714 1/20 0.53
DYRK1A Q13627 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14918157 0.89 HDAC6 (0.71) HDAC6HDAC1HDAC4HDAC8CLK4
SCHEMBL14918305 0.88 HDAC6 (0.69) HDAC6HDAC1HDAC4HDAC8CLK4
SCHEMBL14917912 0.87 HDAC6 (0.59) HDAC6HDAC1HDAC4HDAC8
SCHEMBL14917947 0.85 HDAC6 (0.59) HDAC6HDAC1HDAC4HDAC8
SCHEMBL14918138 0.83 HDAC6 (0.57) HDAC6HDAC1HDAC4HDAC8CLK4
SCHEMBL14918355 0.82 HDAC6 (0.60) HDAC6HDAC1HDAC4HDAC8
SCHEMBL17394582 0.82 HDAC6 (0.56) HDAC6HDAC1HDAC4HDAC8CYP3A4
SCHEMBL14918189 0.80 HDAC6 (0.53) HDAC6HDAC1HDAC4HDAC8CYP3A4
SCHEMBL14918136 0.79 HDAC6 (0.59) HDAC6HDAC1HDAC4HDAC8
SCHEMBL14972195 0.79 CHRNB2 (0.63) HDAC6HDAC1HDAC4HDAC8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013066839-A2 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO claimed
WO-2013066839-A2 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO disclosed