SCHEMBL14920397

SCHEMBL14920397

C[Si](C)(C)C#Cc1ccc(Oc2c(Cl)ccc([CH]CC(N)=O)c2F)cc1

nearest known ligand 0.31

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MET P08581 3/20 0.31
KDR P35968 3/20 0.31
AURKA O14965 1/20 0.31
ABL1 P00519 1/20 0.31
LCK P06239 1/20 0.31
FYN P06241 1/20 0.31
YES1 P07947 1/20 0.31
FGFR2 P21802 1/20 0.31
EPHA2 P29317 1/20 0.31
LTK P29376 1/20 0.31
AXL P30530 1/20 0.31
FLT3 P36888 1/20 0.31
MST1R Q04912 1/20 0.31
PTK6 Q13882 1/20 0.31
HSD17B10 Q99714 1/20 0.30
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14920471 0.81 PARP10 (0.37) HSD17B10
SCHEMBL14920886 0.80 PARP10 (0.43) METKDRAURKAABL1LCK
SCHEMBL14920652 0.80 RAF1 (0.33) HSD17B10
SCHEMBL14920130 0.80 RHEB (0.44) HSD17B10
SCHEMBL14920790 0.77 PTPN7 (0.41)
SCHEMBL14920553 0.76 HSD17B10 (0.43) HSD17B10
SCHEMBL14920459 0.76 LTA4H (0.46)
SCHEMBL14920644 0.76 MAPT (0.37) METKDRAURKAABL1LCK
SCHEMBL14920388 0.74 PPARG (0.34) METKDRAURKAABL1LCK
SCHEMBL14920342 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2773613-A1 SUBSTITUTED BENZYLAMINE COMPOUNDS, THEIR USE IN MEDICINE, AND IN PARTICULAR THE TREATMENT OF HEPATITIS C VIRUS (HCV) INFECTION Astex Therapeutics Limited (GB) 2014-09-10 EP disclosed
WO-2013064538-A1 SUBSTITUTED BENZYLAMINE COMPOUNDS, THEIR USE IN MEDICINE, AND IN PARTICULAR THE TREATMENT OF HEPATITIS C VIRUS (HCV) INFECTION ASTEX THERAPEUTICS LIMITED (GB) 2013-05-10 WO disclosed