SCHEMBL14920799

SCHEMBL14920799

O=C(O)N1CC(CO)C(c2ccc(Cl)cc2)C1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 6/20 0.60
NMT2 O60551 1/20 0.52
CCR5 P51681 1/20 0.46
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14921785 0.87 NMT1 (0.51) NMT1
SCHEMBL14921784 0.87 NMT1 (0.51) NMT1
SCHEMBL14920309 0.87 NMT1 (0.51) NMT1
SCHEMBL4099146 0.86 CCR5 (0.48) NMT1CCR5
SCHEMBL4110254 0.85 NMT1 (0.45) NMT1NMT2CCR5PDE4APDE4B
SCHEMBL20475198 0.85 NMT1 (0.45) NMT1NMT2CCR5CYP1A2CYP3A4
SCHEMBL20475148 0.81 NMT1 (0.57) NMT1NMT2CCR5RECQLPDE4A
SCHEMBL26131609 0.81 KDM1A (0.48) NMT1PDE4APDE4BPDE4CPDE4D
SCHEMBL31412605 0.80 PDE4B (0.59) NMT1NMT2PDE4APDE4BPDE4C
SCHEMBL4011915 0.80 PDE4B (0.59) NMT1NMT2PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2773637-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2014-09-10 EP disclosed
WO-2013064983-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2013-05-10 WO disclosed