SCHEMBL14922151

SCHEMBL14922151

CN(C(=O)c1cccc(CN2Cc3cc(Br)ccc3N=C2N)c1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.57
KDM1A O60341 2/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
MDM2 Q00987 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
ITGB3 P05106 4/20 0.38
ITGA2B P08514 4/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
P2RX7 Q99572 1/20 0.37
PRMT5 O14744 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14922149 0.89 BACE1 (0.56) BACE1KDM1AMAOAMAOBL3MBTL1
SCHEMBL8272691 0.83 BACE1 (0.75) BACE1
SCHEMBL8266893 0.73 BACE1 (0.77) BACE1NPC1RAB9AKMT2A
SCHEMBL5999607 0.73 BACE1 (1.00) BACE1
SCHEMBL14723905 0.72 BACE1 (0.71) BACE1L3MBTL1ALDH1A1SMN1; SMN2NPC1
SCHEMBL6177291 0.70 KDM1A (0.56) KDM1AMAOAMAOBL3MBTL1ALDH1A1
SCHEMBL5350869 0.69 PDE4A (0.48) BACE1
SCHEMBL14723914 0.69 BACE1 (0.69) BACE1
SCHEMBL5999386 0.69 BACE1 (0.72) BACE1
SCHEMBL13525179 0.67 L3MBTL1 (0.57) KDM1AMAOAMAOBL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8436006-B2 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE) JANSSSEN PHARMACEUTICA N.V. (BE) 2013-05-07 US disclosed
US-8436006-B2 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE) JANSSSEN PHARMACEUTICA N.V. (BE) 2013-05-07 US disclosed