SCHEMBL14923948

SCHEMBL14923948

Cc1cc(Nc2nc(N[C@H](CCCNC(=O)OC(C)(C)C)[C@H](C)N)c(F)cc2C(N)=O)cnc1C

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.37
EGFR P00533 2/20 0.37
SYK P43405 4/20 0.35
BRD4 O60885 5/20 0.35
ACVR1B P36896 1/20 0.34
TGFBR1 P36897 1/20 0.34
ACVRL1 P37023 1/20 0.34
STK17B O94768 1/20 0.34
STK17A Q9UEE5 1/20 0.34
MKNK2 Q9HBH9 2/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
STING1 Q86WV6 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14931154 0.92 ITK (0.36) ITKEGFRSYKBRD4ACVR1B
SCHEMBL14923915 0.89 SYK (0.36) SYK
SCHEMBL14923913 0.88 SYK (0.33) ITKEGFRSYKBRD4IRAK4
SCHEMBL14910576 0.87 SYK (0.40) SYK
SCHEMBL14910054 0.86 SYK (0.38) SYK
SCHEMBL16165052 0.86 SYK (0.38) SYK
SCHEMBL14923713 0.86 SYK (0.37) SYK
SCHEMBL14923873 0.86 SYK (0.37) SYK
SCHEMBL14923712 0.85 SYK (0.35) SYK
SCHEMBL16170911 0.85 SYK (0.35) EGFRSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed