SCHEMBL1492989

SCHEMBL1492989

COc1ccccc1NC(=O)Nc1ccc(-c2ccnc(C)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.62
MAPT P10636 4/20 0.60
RAB9A P51151 2/20 0.60
NPC1 O15118 1/20 0.60
PDGFRA P16234 1/20 0.57
KDR P35968 1/20 0.57
PSEN1 P49768 4/20 0.57
PSEN2 P49810 4/20 0.57
APH1B Q8WW43 4/20 0.57
NCSTN Q92542 4/20 0.57
APH1A Q96BI3 4/20 0.57
PSENEN Q9NZ42 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
PORCN Q9H237 1/20 0.57
LMNA P02545 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
ROCK2 O75116 1/20 0.56
LIMK1 P53667 1/20 0.56
AHR P35869 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492687 0.91 PORCN (0.60) SMN1; SMN2MAPTPSEN1PSEN2APH1B
SCHEMBL1492931 0.89 KMT2A (0.65) SMN1; SMN2MAPTRAB9ANPC1PSEN1
SCHEMBL1492959 0.88 PORCN (0.59) PDGFRAKDRPSEN1PSEN2APH1B
SCHEMBL1492881 0.88 PSEN1 (0.56) SMN1; SMN2MAPTRAB9ANPC1PDGFRA
SCHEMBL1492820 0.87 MAPT (0.65) SMN1; SMN2MAPTRAB9AKDRPSEN1
SCHEMBL1492892 0.87 NPC1 (0.55) SMN1; SMN2MAPTRAB9ANPC1PSEN1
SCHEMBL1492794 0.86 PPIA (0.58) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1780926 0.85 PSEN1 (0.61) SMN1; SMN2MAPTRAB9ANPC1PDGFRA
SCHEMBL27809799 0.85 PSEN1 (0.54) SMN1; SMN2MAPTPDGFRAKDRPSEN1
SCHEMBL1493084 0.85 MEN1 (0.58) MAPTRAB9ANPC1PDGFRAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102083794-A Urea compounds as gamma secretase modulators AMGEN INC 2011-06-01 CN claimed
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US claimed
EP-2300427-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2011-03-30 EP claimed
WO-2009137404-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2009-11-12 WO claimed
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US disclosed
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators BACE1, BACE2, PSEN1 SMN1; SMN2 2465/4885MAPT 26/4885RAB9A 1725/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.