SCHEMBL14929923

SCHEMBL14929923

CCCN(C(=O)OC(C)(C)C)c1nc(Nc2cccc(C(=O)OC)c2)c(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.40
MAPK1 P28482 2/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 1/20 0.40
ABCB1 P08183 2/20 0.38
ABCG2 Q9UNQ0 2/20 0.38
PDE5A O76074 1/20 0.38
MAPT P10636 7/20 0.37
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CASR P41180 1/20 0.37
BRD4 O60885 1/20 0.36
EP300 Q09472 1/20 0.36
CREBBP Q92793 1/20 0.36
PDGFRB P09619 1/20 0.36
ROCK1 Q13464 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14923937 0.93 MAPK1 (0.39) TP53MAPK1LMNATSHRABCB1
SCHEMBL14929932 0.78 CAMK1D (0.39) LMNATSHRABCB1ABCG2CDC25B
SCHEMBL14927570 0.76 KHK (0.39) MAPTKDM4EALDH1A1RAB9APOLB
SCHEMBL14929913 0.75 SYK (0.47) ABCB1ABCG2NPC1
SCHEMBL14931174 0.71 CAMK1D (0.39) LMNATSHRABCB1ABCG2CDC25B
SCHEMBL14927585 0.70 ATR (0.36) MAPK1LMNATSHRMAPTKDM4E
SCHEMBL19790365 0.68 TRPA1 (0.39) TP53LMNAABCB1ABCG2MAPT
SCHEMBL14923956 0.68 SYK (0.46) ABCB1ABCG2
SCHEMBL14923933 0.68 KHK (0.38) ALDH1A1
SCHEMBL16169208 0.68 TRPA1 (0.40) TP53ABCB1ABCG2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK TP53 2380/4885MAPK1 334/4885LMNA 3649/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.