SCHEMBL1493023

SCHEMBL1493023

Cc1cc(-c2ccc(NC(=O)Nc3cccc(-c4ccc(F)cc4)c3)cc2)ccn1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.65
PSEN1 P49768 7/20 0.62
PSEN2 P49810 7/20 0.62
APH1B Q8WW43 7/20 0.62
NCSTN Q92542 7/20 0.62
APH1A Q96BI3 7/20 0.62
PSENEN Q9NZ42 7/20 0.62
WNT3A P56704 2/20 0.56
PORCN Q9H237 1/20 0.56
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TP53 P04637 2/20 0.53
POLB P06746 1/20 0.52
KMT2A Q03164 1/20 0.52
MGLL Q99685 1/20 0.51
GBA1 P04062 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492826 0.94 PSEN1 (0.61) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492821 0.91 PSEN1 (0.63) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1492860 0.90 CNR1 (0.68) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492870 0.86 PSEN1 (0.67) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492983 0.86 PORCN (0.69) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1493028 0.86 PSEN1 (0.68) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492874 0.85 CNR1 (0.65) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492772 0.85 PSEN1 (0.69) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1492858 0.85 CNR1 (0.65) CNR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1493038 0.85 PSEN1 (0.71) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US claimed
EP-2300427-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2011-03-30 EP claimed
WO-2009137404-A1 UREA COMPOUNDS AS GAMMA SECRETASE MODULATORS AMGEN INC. (US) 2009-11-12 WO claimed
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US disclosed
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators AMGEN INC. 2011-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118234-A1 Urea Compounds as Gamma Secretase Modulators BACE1, BACE2, PSEN1 CNR1 2240/4885PSEN1 3/4885PSEN2 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.