SCHEMBL14932001

SCHEMBL14932001

NC(=O)Oc1cnc(-n2ncc3c(N)ncnc32)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 7/20 0.48
KDM4E B2RXH2 3/20 0.45
PI4KA P42356 2/20 0.45
PI4K2B Q8TCG2 2/20 0.45
PI4K2A Q9BTU6 2/20 0.45
PI4KB Q9UBF8 2/20 0.45
HSD17B10 Q99714 2/20 0.45
EGFR P00533 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
TSHR P16473 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
RAB9A P51151 5/20 0.40
NPC1 O15118 4/20 0.40
HTT P42858 1/20 0.40
BLM P54132 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14931966 0.90 XDH (0.51) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL14932063 0.87 XDH (0.47) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3868155 0.81 XDH (0.51) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL14932046 0.79 XDH (0.49) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3872178 0.79 XDH (0.57) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3878342 0.78 XDH (0.48) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3868852 0.77 XDH (0.49) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3878769 0.76 XDH (0.51) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3878745 0.74 XDH (0.54) XDHKDM4EPI4KAPI4K2BPI4K2A
SCHEMBL3878154 0.72 XDH (0.49) XDHKDM4EPI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827444-B1 MNK1 OR MNK2 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2013-05-15 EP claimed