SCHEMBL14939119

SCHEMBL14939119

CCc1ccccc1CN1CCN(C2(c3cccc(N4CCN(C)CC4)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.51
NPSR1 Q6W5P4 1/20 0.50
HTR7 P34969 4/20 0.47
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HRH2 P25021 1/20 0.41
DRD3 P35462 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
HTR1A P08908 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939868 0.92 NPSR1 (0.52) MAPTNPSR1HTR7LMNATP53
SCHEMBL14940024 0.91 MAPT (0.50) MAPTNPSR1HTR7LMNATP53
SCHEMBL14939311 0.91 NPSR1 (0.51) MAPTNPSR1HTR7LMNATP53
SCHEMBL14939938 0.89 MAPT (0.51) MAPTNPSR1HTR7LMNADRD2
SCHEMBL14939603 0.89 NPSR1 (0.49) MAPTNPSR1HTR7LMNATP53
SCHEMBL14940181 0.88 NPSR1 (0.67) MAPTNPSR1HTR7LMNADRD2
SCHEMBL14939507 0.85 MAPT (0.48) MAPTNPSR1HTR7LMNATP53
SCHEMBL14940061 0.84 NPSR1 (0.57) MAPTNPSR1HTR7LMNATP53
SCHEMBL14939809 0.83 NPSR1 (0.51) MAPTNPSR1HTR7LMNATP53
SCHEMBL14939244 0.83 NPSR1 (0.71) MAPTNPSR1HTR7LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed