SCHEMBL14939167

SCHEMBL14939167

COc1cccc2c1C(=O)C(c1ccccc1)(N1CCN(Cc3ccccc3)CC1)C2=O

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.70
MAPT P10636 2/20 0.49
MMP2 P08253 2/20 0.47
MMP9 P14780 2/20 0.47
UTS2R Q9UKP6 1/20 0.45
ACHE P22303 1/20 0.45
LMNA P02545 1/20 0.44
SIGMAR1 Q99720 3/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTR7 P34969 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940444 0.88 NPSR1 (0.53) NPSR1MAPTACHELMNAALDH1A1
SCHEMBL14939694 0.84 NPSR1 (0.73) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14940046 0.84 NPSR1 (0.54) NPSR1MAPTLMNAALDH1A1MEN1
SCHEMBL14939688 0.84 NPSR1 (0.77) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14939617 0.83 NPSR1 (1.00) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14939390 0.83 NPSR1 (0.75) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14939436 0.83 NPSR1 (0.61) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14939775 0.83 NPSR1 (0.52) NPSR1MAPTALDH1A1MEN1KMT2A
SCHEMBL14939178 0.82 NPSR1 (0.77) NPSR1MAPTMMP2MMP9LMNA
SCHEMBL14939174 0.82 NPSR1 (0.65) NPSR1MAPTLMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed