SCHEMBL14939445

SCHEMBL14939445

CCc1ccccc1CN1CCN(C2(c3cc(C)cc(OC)c3)C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.51
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 6/20 0.47
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
HTR7 P34969 3/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
ALOX15 P16050 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939336 0.94 NPSR1 (0.52) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939573 0.92 TP53 (0.51) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939199 0.90 NPSR1 (0.55) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939824 0.90 NPSR1 (0.49) TP53NPSR1MAPTALDH1A1HTR7
SCHEMBL14938832 0.89 NPSR1 (0.47) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939200 0.88 NPSR1 (0.53) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939326 0.88 NPSR1 (0.65) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14940020 0.86 NPSR1 (0.51) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939859 0.85 TP53 (0.49) TP53NPSR1MAPTALDH1A1KDM4E
SCHEMBL14939296 0.85 NPSR1 (0.50) TP53NPSR1MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed