SCHEMBL14939573

SCHEMBL14939573

COc1cc(C)cc(C2(N3CCN(Cc4ccccc4C)CC3)C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.51
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 4/20 0.47
LMNA P02545 3/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KMT2A Q03164 1/20 0.41
HTT P42858 1/20 0.41
HTR7 P34969 1/20 0.40
ACHE P22303 2/20 0.39
CYP2A13 Q16696 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940020 0.95 NPSR1 (0.51) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939445 0.92 TP53 (0.51) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939539 0.90 NPSR1 (0.55) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939824 0.90 NPSR1 (0.49) TP53NPSR1MAPTALDH1A1KMT2A
SCHEMBL14939490 0.90 TP53 (0.47) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939859 0.89 TP53 (0.49) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939577 0.89 NPSR1 (0.52) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939326 0.88 NPSR1 (0.65) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939001 0.87 TP53 (0.60) TP53NPSR1MAPTLMNAKDM4E
SCHEMBL14939725 0.86 TP53 (0.47) TP53NPSR1MAPTLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed