SCHEMBL14939690

SCHEMBL14939690

O=C1c2ccccc2C(=O)C1(c1cccnc1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.77
CHRM2 P08172 2/20 0.46
CHRM3 P20309 1/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
DHPS P49366 2/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
KDM4E B2RXH2 1/20 0.45
TRPV6 Q9H1D0 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940290 0.90 NPSR1 (0.63) NPSR1CHRM2CHRM3ALDH1A1MAPT
SCHEMBL14939850 0.88 NPSR1 (0.60) NPSR1CHRM2CHRM3ALDH1A1LMNA
SCHEMBL14939391 0.88 NPSR1 (0.60) NPSR1ALDH1A1TP53MAPTRAB9A
SCHEMBL14939617 0.87 NPSR1 (1.00) NPSR1LMNAMAPTMMP2MMP9
SCHEMBL14939742 0.86 NPSR1 (0.82) NPSR1LMNAMAPTMMP2MMP9
SCHEMBL14940333 0.86 NPSR1 (0.57) NPSR1CHRM3ALDH1A1MAPTMAPK1
SCHEMBL14940026 0.86 NPSR1 (0.56) NPSR1CHRM2CHRM3ALDH1A1MAPT
SCHEMBL14939499 0.85 NPSR1 (0.55) NPSR1CHRM2CHRM3ALDH1A1LMNA
SCHEMBL14938982 0.84 NPSR1 (0.64) NPSR1CHRM2CHRM3ALDH1A1LMNA
SCHEMBL14939951 0.84 NPSR1 (0.54) NPSR1ALDH1A1LMNAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed