SCHEMBL14938982

SCHEMBL14938982

O=C1c2cccc(Cl)c2C(=O)C1(c1ccccc1)N1CCN(Cc2cccnc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.64
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
TRPV6 Q9H1D0 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
OPRL1 P41146 1/20 0.42
P2RX7 Q99572 2/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939688 0.91 NPSR1 (0.77) NPSR1DRD2DRD4DRD3LMNA
SCHEMBL14939243 0.90 NPSR1 (0.65) NPSR1ALDH1A1KDM4EOPRL1LMNA
SCHEMBL14939115 0.88 NPSR1 (0.60) NPSR1TRPV6CHRM2CHRM3ALDH1A1
SCHEMBL14939690 0.84 NPSR1 (0.77) NPSR1TRPV6CHRM2CHRM3ALDH1A1
SCHEMBL14939318 0.82 NPSR1 (0.60) NPSR1DRD2DRD4DRD3TRPV6
SCHEMBL14939436 0.81 NPSR1 (0.61) NPSR1CHRM2CHRM3ALDH1A1KDM4E
SCHEMBL14940290 0.80 NPSR1 (0.63) NPSR1DRD2TRPV6CHRM2CHRM3
SCHEMBL14939617 0.79 NPSR1 (1.00) NPSR1DRD2LMNAMAPTMMP2
SCHEMBL14939390 0.79 NPSR1 (0.75) NPSR1DRD2OPRM1LMNAMAPT
SCHEMBL14939299 0.79 NPSR1 (0.58) NPSR1ALDH1A1KDM4EP2RX7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed