SCHEMBL14940323

SCHEMBL14940323

COc1cccc(C2(N3CCN(Cc4ccc(C)cc4C)CC3)C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.54
NPSR1 Q6W5P4 1/20 0.49
MAPT P10636 4/20 0.47
LMNA P02545 1/20 0.43
GRIN2B Q13224 2/20 0.41
HTR7 P34969 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939577 0.91 NPSR1 (0.52) TP53NPSR1MAPTLMNAHTR7
SCHEMBL14939514 0.90 NPSR1 (0.47) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14939110 0.90 NPSR1 (0.55) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14939200 0.88 NPSR1 (0.53) TP53NPSR1MAPTLMNAHTR7
SCHEMBL14939486 0.88 TP53 (0.52) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14939106 0.88 NPSR1 (0.64) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14939761 0.87 NPSR1 (0.61) TP53NPSR1MAPTSIGMAR1DRD2
SCHEMBL14939396 0.86 NPSR1 (0.51) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14940165 0.86 NPSR1 (0.51) TP53NPSR1MAPTLMNAGRIN2B
SCHEMBL14940141 0.86 NPSR1 (0.54) TP53NPSR1MAPTLMNAGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed