SCHEMBL14943013

SCHEMBL14943013

CCCOc1ccc2sc(S(=O)(=O)NCP(=O)(O)Oc3ccc(C#N)c(C(F)(F)F)c3)cc2c1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.36
PLA2G7 Q13093 1/20 0.35
CLK1 P49759 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14943012 0.94 AR (0.36) ARPLA2G7
SCHEMBL13032081 0.93 TRPV4 (0.36) ARPLA2G7
SCHEMBL14931299 0.90 AR (0.32) ARPLA2G7
SCHEMBL14943014 0.90 AR (0.36) ARPLA2G7
SCHEMBL16684156 0.89 TRPV4 (0.34) ARPLA2G7
SCHEMBL14943020 0.89 TRPV4 (0.34) ARPLA2G7
SCHEMBL14943032 0.89 TRPV4 (0.37)
SCHEMBL14943071 0.89 AR (0.36) ARPLA2G7
SCHEMBL16684163 0.88 AR (0.33) AR
SCHEMBL14943084 0.88 AR (0.35) ARPLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8440643-B2 Inhibitors of beta-lactamase METHYLGENE INC. (CA) 2013-05-14 US disclosed