SCHEMBL14944179

SCHEMBL14944179

COc1cccc(Oc2ccc(-c3cc(C(F)(F)F)c(C#N)c(=O)n3Cc3ccc(C)cc3C)cc2C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.51
NR1H3 Q13133 4/20 0.51
RXRA P19793 3/20 0.51
KDM4E B2RXH2 2/20 0.41
GLA P06280 2/20 0.41
GAA P10253 2/20 0.41
ALDH1A1 P00352 1/20 0.41
AR P10275 8/20 0.38
MEN1 O00255 1/20 0.38
CNR1 P21554 1/20 0.38
GPR183 P32249 1/20 0.38
CNR2 P34972 1/20 0.38
KMT2A Q03164 1/20 0.38
PGR P06401 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPT P10636 2/20 0.36
NAAA Q02083 1/20 0.35
FFAR1 O14842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2386372 0.93 NR1H2 (0.52) NR1H2NR1H3RXRAARMEN1
SCHEMBL2388648 0.93 RXRA (0.53) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2389162 0.92 NR1H2 (0.51) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2391088 0.91 NR1H2 (0.51) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2263493 0.91 NR1H2 (0.62) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2389952 0.90 NR1H2 (0.48) NR1H2NR1H3RXRAARMEN1
SCHEMBL2262770 0.90 NR1H2 (0.53) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2387552 0.90 NR1H2 (0.52) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2387075 0.90 NR1H2 (0.49) NR1H2NR1H3RXRAKDM4EGLA
SCHEMBL2385089 0.89 NR1H2 (0.51) NR1H2NR1H3RXRAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465869-B1 MODULATORS OF LXR EXELIXIS PATENT CO LLC (US) 2013-05-15 EP disclosed