SCHEMBL14944714

SCHEMBL14944714

COC(=O)c1cccc(Cn2c(=O)n(N)c3c(N)nc(-n4cccn4)nc32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.44
ABHD6 Q9BV23 1/20 0.41
ADORA2A P29274 4/20 0.39
ADORA1 P30542 3/20 0.39
TPH1 P17752 2/20 0.39
TPH2 Q8IWU9 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
IDO1 P14902 1/20 0.39
YTHDC1 Q96MU7 1/20 0.39
MAPK10 P53779 1/20 0.38
TSHR P16473 1/20 0.38
MAPK8 P45983 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
OPRD1 P41143 1/20 0.37
F10 P00742 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944673 0.83 TLR7 (0.64) TLR7ADORA1
SCHEMBL21581161 0.75 TLR7 (0.55) TLR7ADORA1
SCHEMBL20343835 0.75 TLR7 (0.40) TLR7ABHD6ADORA2AADORA1LOXL2
SCHEMBL21581162 0.73 TLR7 (0.51) TLR7ADORA1
SCHEMBL19423866 0.73 TLR7 (0.63) TLR7
SCHEMBL14944641 0.72 TLR7 (0.50) TLR7ADORA1
SCHEMBL20343750 0.69 LOXL2 (0.38) TLR7ADORA2AADORA1LOXL2YTHDC1
SCHEMBL14987126 0.69 HTT (0.71) ABHD6LOXL2IDO1MAPK10TSHR
SCHEMBL19423908 0.69 TLR7 (0.50) TLR7ADORA1
SCHEMBL14944614 0.67 TLR7 (0.51) TLR7ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068438-A1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN R&D IRELAND (IE) 2013-05-16 WO disclosed