SCHEMBL14949225

SCHEMBL14949225

CSc1nc(N)cc(Oc2ccc(-c3cnc(Nc4cccc(C)c4)[nH]3)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.51
KIT P10721 1/20 0.51
PDGFRA P16234 1/20 0.51
CDK11B P21127 1/20 0.51
FLT3 P36888 1/20 0.51
CDKL2 Q92772 1/20 0.51
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HTT P42858 1/20 0.37
CDK8 P49336 2/20 0.37
LMNA P02545 3/20 0.36
RXFP1 Q9HBX9 1/20 0.36
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
EGFR P00533 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625061 0.89 PDGFRB (0.67) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL12336289 0.84 PDGFRB (0.56) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL17658742 0.81 PDGFRB (0.42) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL14949396 0.78 PDGFRB (0.51) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL14949579 0.77 PDGFRB (0.48) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL13547695 0.77 PDGFRB (0.50) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL14949269 0.76 PDGFRB (0.47) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL627644 0.76 PDGFRB (0.50) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL14949294 0.76 KIT (0.47) PDGFRBKITPDGFRACDK11BFLT3
SCHEMBL14949283 0.76 PDGFRB (0.45) PDGFRBKITPDGFRACDK11BFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2016-04-07 US disclosed
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2015-06-11 US disclosed
US-8957216-B2 Heterocyclic compounds useful for kinase inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. (US) 2015-02-17 US disclosed
US-20130266636-A1 METHODS FOR BLOCKING CELL PROLIFERATION AND TREATING DISEASES AND CONDITIONS RESPONSIVE TO CELL GROWTH INHIBITION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-10-10 US disclosed
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION AMITECH THERAPEUTIC SOLUTIONS INC (US) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION MAP4K2, MAP3K20, MAP3K19 PDGFRB 497/4885KIT 540/4885PDGFRA 498/4885
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 PDGFRB 497/4885KIT 540/4885PDGFRA 498/4885
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 PDGFRB 497/4885KIT 540/4885PDGFRA 498/4885
US-20130266636-A1 METHODS FOR BLOCKING CELL PROLIFERATION AND TREATING DISEASES AND CONDITIONS RESPONSIVE TO CELL GROWTH INHIBITION BRAF, BUB1B, MKI67 PDGFRB 1405/4885KIT 1806/4885PDGFRA 1972/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.