SCHEMBL14949672

SCHEMBL14949672

O=C(O)Nc1ccc(Oc2ccc([N+](=O)[O-])cn2)c(F)c1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 3/20 0.67
MET P08581 2/20 0.49
MAPT P10636 7/20 0.46
MEN1 O00255 6/20 0.46
KMT2A Q03164 6/20 0.46
PABPC1 P11940 3/20 0.45
POLB P06746 2/20 0.45
L3MBTL1 Q9Y468 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 1/20 0.44
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RAF1 P04049 1/20 0.43
KDM4E B2RXH2 2/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14949670 1.00 HSPB1 (0.67) HSPB1METMAPTMEN1KMT2A
SCHEMBL2859670 0.91 HSPB1 (0.57) HSPB1METMAPTMEN1KMT2A
SCHEMBL2859667 0.91 HSPB1 (0.57) HSPB1METMAPTMEN1KMT2A
SCHEMBL12469298 0.87 HSPB1 (0.52) HSPB1MAPTMEN1KMT2APABPC1
SCHEMBL12469297 0.87 HSPB1 (0.52) HSPB1MAPTMEN1KMT2APABPC1
SCHEMBL15301357 0.85 MAPT (0.55) HSPB1MAPTMEN1KMT2APABPC1
SCHEMBL15301358 0.85 MAPT (0.55) HSPB1MAPTMEN1KMT2APABPC1
SCHEMBL12892603 0.85 HSPB1 (0.59) HSPB1METMAPTMEN1KMT2A
SCHEMBL2851303 0.85 HSPB1 (0.49) HSPB1MAPTMEN1KMT2APABPC1
SCHEMBL2851309 0.85 HSPB1 (0.49) HSPB1MAPTMEN1KMT2APABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445509-B2 Fused heterocyclic derivatives and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-21 US disclosed