SCHEMBL14949679

SCHEMBL14949679

O=C(O)Nc1ccc(Oc2ccc3nc(NC(=O)C4CC4)cn3c2)c(F)c1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.70
MET P08581 9/20 0.70
FLT1 P17948 2/20 0.67
FLT4 P35916 1/20 0.67
AURKA O14965 1/20 0.53
PDGFRB P09619 1/20 0.53
KIT P10721 1/20 0.53
LRRK2 Q5S007 2/20 0.50
BRAF P15056 3/20 0.49
ABL1 P00519 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447930 0.95 KDR (0.70) KDRMETFLT1FLT4AURKA
SCHEMBL1258959 0.87 KDR (0.65) KDRMETFLT1FLT4AURKA
SCHEMBL12892681 0.86 KDR (0.65) KDRMETFLT1FLT4AURKA
Hydrochloric Acid SCHEMBL1260024 0.86 KDR (0.65) KDRMETFLT1FLT4AURKA
SCHEMBL1257985 0.86 KDR (0.59) KDRMETFLT1FLT4AURKA
SCHEMBL1260492 0.86 MET (0.60) KDRMETFLT1FLT4AURKA
SCHEMBL14949677 0.86 KDR (0.58) KDRMETFLT1FLT4AURKA
SCHEMBL1259967 0.83 MET (1.00) KDRMETFLT1FLT4AURKA
SCHEMBL1259136 0.83 KDR (0.56) KDRMETFLT1FLT4AURKA
Hydrochloric Acid SCHEMBL29363414 0.83 MET (1.00) KDRMETFLT1FLT4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445509-B2 Fused heterocyclic derivatives and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-21 US disclosed