SCHEMBL14960370

SCHEMBL14960370

Cc1nc2ccc(-c3ccc4c(c3)CN(C(=O)N3CCC(CCc5ccc(Cl)cc5)CC3)CCO4)cc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 14/20 0.56
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
CREBBP Q92793 1/20 0.39
RIPK1 Q13546 1/20 0.38
CHEK2 O96017 1/20 0.37
FAAH O00519 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724278 0.92 PIK3CA (0.56) PIK3CACREBBP
SCHEMBL3798408 0.88 PIK3CA (0.62) PIK3CABCHEACHECREBBP
SCHEMBL3795779 0.87 PIK3CA (0.60) PIK3CABCHEACHECREBBP
SCHEMBL3788978 0.87 PIK3CA (0.61) PIK3CACREBBP
SCHEMBL3793252 0.86 PIK3CA (0.62) PIK3CACREBBP
SCHEMBL2724447 0.85 PIK3CA (0.56) PIK3CACREBBPCHEK2
SCHEMBL6126859 0.85 PIK3CA (0.57) PIK3CABCHEACHE
SCHEMBL3799035 0.84 PIK3CA (0.61) PIK3CACREBBPRIPK1
SCHEMBL3794536 0.84 PIK3CA (0.64) PIK3CACREBBP
SCHEMBL2725831 0.84 PIK3CA (0.64) PIK3CACREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2435426-B1 BENZOXAZEPINES AS INHIBITORS OF PI3K/m TOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS INC (US) 2013-05-22 EP disclosed