SCHEMBL14965241

SCHEMBL14965241

c1ccc(-c2csc3ncnc(NC4CCNCC4)c23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 6/20 0.53
LMNA P02545 7/20 0.52
MAPK1 P28482 3/20 0.52
HTT P42858 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
TNF P01375 1/20 0.51
NOD1 Q9Y239 1/20 0.51
ADRB3 P13945 1/20 0.51
CSNK2A2 P19784 2/20 0.50
CSNK2B P67870 2/20 0.50
CSNK2A1 P68400 2/20 0.50
THRB P10828 1/20 0.50
PTPN5 P54829 1/20 0.50
DAPK3 O43293 1/20 0.50
PRKD3 O94806 1/20 0.50
MAP4K4 O95819 1/20 0.50
ABL1 P00519 1/20 0.50
NTRK1 P04629 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965340 0.88 LMNA (0.52) FGFR1LMNAHTTSMN1; SMN2MEN1
SCHEMBL14965085 0.88 FGFR1 (0.53) FGFR1LMNAHTTSMN1; SMN2MEN1
SCHEMBL2368170 0.88 FGFR1 (0.55) FGFR1LMNAMAPK1HTTSMN1; SMN2
SCHEMBL13319858 0.87 FGFR1 (0.57) FGFR1LMNAMAPK1HTTSMN1; SMN2
SCHEMBL6642610 0.83 FGFR1 (0.55) FGFR1LMNAMAPK1HTTSMN1; SMN2
SCHEMBL1606116 0.80 LMNA (0.76) LMNAMAPK1HTTSMN1; SMN2MEN1
SCHEMBL31462338 0.79 FGFR1 (0.53) FGFR1LMNAMAPK1HTTSMN1; SMN2
SCHEMBL14965069 0.79 IRAK4 (0.69) LMNAHTTSMN1; SMN2MEN1KMT2A
SCHEMBL5671622 0.78 LRRK2 (0.56) FGFR1MAPK1MEN1KMT2APRKD3
SCHEMBL14965213 0.77 FGFR1 (0.55) FGFR1LMNAMAPK1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP claimed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO claimed
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP disclosed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO disclosed