SCHEMBL14965339

SCHEMBL14965339

CN(C)C1CCN(c2ncnc3scc(-c4ccccc4)c23)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.67
ADRB3 P13945 2/20 0.66
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16292947 0.94 ADRB3 (0.60) LMNAADRB3
SCHEMBL16292822 0.91 ADRB3 (0.60) ADRB3
SCHEMBL17599009 0.87 ADRB3 (0.58) ADRB3
SCHEMBL24391624 0.87 ADRB3 (0.59) LMNAADRB3MEN1KMT2A
SCHEMBL14964948 0.87 ADRB3 (0.59) LMNAADRB3KMT2A
SCHEMBL4432115 0.85 LMNA (0.72) LMNAMEN1KMT2A
SCHEMBL4552668 0.85 LMNA (0.72) LMNAMEN1KMT2A
SCHEMBL16294397 0.85 LMNA (0.72) LMNAMEN1KMT2A
SCHEMBL16293493 0.84 ADRB3 (0.64) ADRB3KMT2A
SCHEMBL14965408 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780343-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS Xention Limited (GB) 2014-09-24 EP disclosed
CN-104011054-A Thieno- and furo-pyrimidines and pyridines, useful as potassium channel inhibitors XENTION LTD 2014-08-27 CN disclosed
WO-2013072694-A1 THIENO- AND FURO - PYRIMIDINES AND PYRIDINES, USEFUL AS POTASSIUM CHANNEL INHIBITORS XENTION LIMITED (GB) 2013-05-23 WO disclosed