SCHEMBL14965624

SCHEMBL14965624

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccc(-c3ccc(OC(F)(F)F)cc3)cc1)CC2

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.57
KCNH2 Q12809 5/20 0.51
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
PTGS1 P23219 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
DRD4 P21917 3/20 0.39
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
KCNJ1 P48048 1/20 0.38
STAT3 P40763 2/20 0.38
TEAD1 P28347 2/20 0.38
GRM2 Q14416 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
LSS P48449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965842 0.97 CHRM1 (0.59) CHRM1KCNH2ALDH1A1TSHRPTGS1
SCHEMBL14966124 0.92 CHRM1 (0.54) CHRM1KCNH2ALDH1A1TSHRPTGS1
SCHEMBL14965658 0.91 CHRM1 (0.48) CHRM1KCNH2ALDH1A1TSHRPTGS1
SCHEMBL14966083 0.90 CHRM1 (0.52) CHRM1KCNH2ALDH1A1TSHRPTGS1
SCHEMBL14966106 0.88 SMN1; SMN2 (0.46) CHRM1KCNH2ALDH1A1TSHRDRD4
SCHEMBL14965750 0.88 CHKA (0.43) CHRM1KCNH2ALDH1A1KCNJ1
SCHEMBL14965483 0.87 CHRM1 (0.49) CHRM1KCNH2ALDH1A1TSHRPTGS1
SCHEMBL14965959 0.87 KCNH2 (0.53) CHRM1KCNH2ALDH1A1TSHRSTAT3
SCHEMBL14965737 0.87 CHRM1 (0.49) CHRM1KCNH2ALDH1A1TSHR
SCHEMBL14966147 0.87 KCNH2 (0.53) CHRM1KCNH2ALDH1A1TSHRSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed