SCHEMBL14965737

SCHEMBL14965737

O=C(NCc1ccc(OC(F)(F)F)cc1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.49
TSHR P16473 1/20 0.47
KCNH2 Q12809 5/20 0.45
HDAC4 P56524 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
EPHX2 P34913 3/20 0.44
NR1H4 Q96RI1 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CHRM2 P08172 1/20 0.42
NAMPT P43490 1/20 0.41
ABL1 P00519 1/20 0.41
MLLT1 Q03111 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
PTGER4 P35408 2/20 0.40
HTR2C P28335 1/20 0.40
SCN3A Q9NY46 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965591 0.92 CHRM3 (0.47) CHRM1TSHRKCNH2HDAC4HDAC6
SCHEMBL14965959 0.91 KCNH2 (0.53) CHRM1TSHRKCNH2ALDH1A1ABL1
SCHEMBL14966147 0.91 KCNH2 (0.53) CHRM1TSHRKCNH2ALDH1A1ABL1
SCHEMBL14965538 0.90 HDAC4 (0.49) TSHRHDAC4HDAC6ALDH1A1MLLT1
SCHEMBL14965611 0.90 TSHR (0.61) TSHRHDAC4HDAC6EPHX2NR1H4
SCHEMBL14966124 0.89 CHRM1 (0.54) CHRM1TSHRKCNH2ALDH1A1NAMPT
SCHEMBL14965842 0.89 CHRM1 (0.59) CHRM1TSHRKCNH2ALDH1A1ABL1
SCHEMBL14965754 0.89 TSHR (0.47) CHRM1TSHRHDAC4HDAC6ALDH1A1
SCHEMBL14965800 0.88 ALDH1A1 (0.58) TSHRKCNH2HDAC4HDAC6ALDH1A1
SCHEMBL14965548 0.87 CHRM1 (0.52) CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed