SCHEMBL14966858

SCHEMBL14966858

Cc1cc([C@H](C)Oc2ccccc2)ccc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
LTB4R Q15722 6/20 0.45
LTB4R2 Q9NPC1 6/20 0.45
ALOX5 P09917 1/20 0.45
FFAR1 O14842 1/20 0.43
IGLV6-57 P01721 1/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
NR1H4 Q96RI1 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18703603 1.00 ALDH1A1 (0.45) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL19193471 1.00 ALDH1A1 (0.45) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL14972264 0.87 TSHR (0.48) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL19194090 0.87 TSHR (0.48) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL14967139 0.87 TSHR (0.48) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL14966804 0.84 TSHR (0.45) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL14966813 0.84 FFAR1 (0.46) ALDH1A1LTB4RLTB4R2ALOX5FFAR1
SCHEMBL10417835 0.81 AKR1C2 (0.51) ALDH1A1KMT2AMEN1RXRARXRB
SCHEMBL14968952 0.80 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1RXRARXRB
SCHEMBL14967524 0.79 KMT2A (0.59) LTB4RLTB4R2ALOX5FFAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9206128-B2 Modulators of methyl modifying enzymes, compositions and uses thereof CONSTELLATION PHARMACEUTICALS, INC. (US) 2015-12-08 US disclosed
US-9206128-B2 Modulators of methyl modifying enzymes, compositions and uses thereof CONSTELLATION PHARMACEUTICALS, INC. (US) 2015-12-08 US disclosed
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed