SCHEMBL14966924

SCHEMBL14966924

Cc1cc(C)c(CNC(=O)c2ccc(C(C)Oc3ccccc3I)c(F)c2)c(O)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 14/20 0.37
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.35
ROS1 P08922 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966641 0.88 SMN1; SMN2 (0.40) KLKB1MAPTSMN1; SMN2TP53
SCHEMBL14967162 0.88 SMN1; SMN2 (0.40) KLKB1MAPTSMN1; SMN2TP53
SCHEMBL14967484 0.88 SMN1; SMN2 (0.40) KLKB1MAPTSMN1; SMN2TP53
SCHEMBL14969791 0.81 TDP1 (0.39) KLKB1MAPTSMN1; SMN2ROS1LMNA
SCHEMBL14969477 0.81 TDP1 (0.39) KLKB1MAPTSMN1; SMN2ROS1LMNA
SCHEMBL14966934 0.81 TDP1 (0.39) KLKB1MAPTSMN1; SMN2ROS1LMNA
SCHEMBL14967045 0.80 SMN1; SMN2 (0.41) KLKB1MAPTSMN1; SMN2TP53LMNA
SCHEMBL14966826 0.80 SMN1; SMN2 (0.41) KLKB1MAPTSMN1; SMN2TP53LMNA
SCHEMBL14966473 0.78 MAPK14 (0.42) KLKB1MAPTSMN1; SMN2TP53ROS1
SCHEMBL14967281 0.78 KDM4E (0.41) KLKB1MAPTSMN1; SMN2TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed