SCHEMBL14967159

SCHEMBL14967159

COC(=O)c1cc(Br)c(C(C)=O)nc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 6/20 0.41
HPGD P15428 3/20 0.41
GAA P10253 4/20 0.38
HSD17B10 Q99714 3/20 0.38
GLA P06280 2/20 0.38
MAPT P10636 2/20 0.38
TSHR P16473 2/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
ATM Q13315 1/20 0.38
SOS1 Q07889 1/20 0.38
CFTR P13569 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
CYP2C9 P11712 1/20 0.37
ABL1 P00519 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21875403 0.81 ALDH1A1 (0.47) KDM4EALDH1A1HPGDGAAHSD17B10
Acetic Acid SCHEMBL29164016 0.80 ALDH1A1 (0.43) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL29824155 0.79 KDM4E (0.44) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL25360368 0.79 KDM4E (0.44) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL2013864 0.77 NPSR1 (0.47) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL30500676 0.76 SOS1 (0.48) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL25262355 0.76 SOS1 (0.48) KDM4EALDH1A1HPGDMAPTTSHR
Trifluoroacetic Acid SCHEMBL25305646 0.76 SOS1 (0.42) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL25360143 0.75 GAA (0.41) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL27388974 0.74 NPSR1 (0.44) KDM4EALDH1A1HPGDGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed