SCHEMBL14968925

SCHEMBL14968925

CC(C)[C@H](OC(N)=O)C(=O)N1CCC[C@H]1c1nc2c(ccc3c4c(ccc32)-c2ccc(B3OC(C)(C)C(C)(C)O3)cc2CO4)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.34
HCRTR1 O43613 9/20 0.33
HCRTR2 O43614 9/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979776 0.87 CYP3A4 (0.46)
SCHEMBL6126547 0.87 CYP3A4 (0.38) HCRTR1HCRTR2
SCHEMBL15052198 0.87 HCRTR1 (0.35) PARP1HCRTR1HCRTR2
SCHEMBL21330022 0.87 CYP3A4 (0.38) HCRTR1HCRTR2
SCHEMBL6126614 0.87 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL19528097 0.85 CYP3A4 (0.44)
SCHEMBL14979634 0.85 PTGES (0.37) PARP1HCRTR1HCRTR2
SCHEMBL8752362 0.79 CYP3A4 (0.44)
SCHEMBL14979730 0.78 CYP3A4 (0.45)
SCHEMBL22364713 0.77 CYP3A4 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635588-A1 CONDENSED IMIDAZOLYLIMIDAZOLES AS ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2013-09-11 EP disclosed
WO-2013075029-A1 CONDENSED IMIDAZOLYLIMIDAZOLES AS ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2013-05-23 WO disclosed