SCHEMBL14968982

SCHEMBL14968982

NC(=O)c1cc2c(OCCO)c(Br)c(C(F)(F)F)nc2nc1N

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
EEF2K O00418 1/20 0.32
PDK2 Q15119 1/20 0.32
KDM4E B2RXH2 2/20 0.31
DHPS P49366 2/20 0.31
S1PR1 P21453 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969047 0.81 EEF2K (0.34) IDO1EEF2KIKBKB
SCHEMBL14969144 0.81 EEF2K (0.35) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14969004 0.80 IKBKB (0.36) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14969024 0.79 RCE1 (0.36) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14969265 0.78 KDM4E (0.35) IDO1EEF2KKDM4EALDH1A1HPGD
SCHEMBL14968912 0.78 RCE1 (0.38) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14969095 0.78 ENPP1 (0.40) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14968979 0.77 IDO1 (0.36) IDO1EEF2KKDM4EALDH1A1GLA
SCHEMBL14969029 0.77 LRRK2 (0.33) IDO1EEF2KKDM4EALDH1A1HPGD
SCHEMBL14969252 0.75 EEF2K (0.34) IDO1EEF2KKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed