SCHEMBL14969024

SCHEMBL14969024

NC(=O)c1cc2c(O)c(Br)c(C(F)(F)F)nc2nc1N

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RCE1 Q9Y256 1/20 0.36
IDO1 P14902 1/20 0.36
IKBKB O14920 1/20 0.35
EEF2K O00418 3/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CD38 P28907 1/20 0.31
EEF2 P13639 1/20 0.31
TBK1 Q9UHD2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14968912 0.88 RCE1 (0.38) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14969004 0.88 IKBKB (0.36) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14969095 0.86 ENPP1 (0.40) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14969144 0.84 EEF2K (0.35) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14969252 0.83 EEF2K (0.34) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14969047 0.82 EEF2K (0.34) RCE1IDO1IKBKBEEF2KEEF2
SCHEMBL14968979 0.80 IDO1 (0.36) RCE1IDO1IKBKBEEF2KKDM4E
SCHEMBL14968982 0.79 IDO1 (0.33) IDO1IKBKBEEF2KKDM4EALDH1A1
SCHEMBL14969265 0.79 KDM4E (0.35) IDO1IKBKBEEF2KKDM4EALDH1A1
SCHEMBL14969228 0.77 GAA (0.33) IDO1IKBKBEEF2KGAACD38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072882-A1 2 -AMINO- 1, 8 -NAPHTHYRIDINE-3 -CARBOXAMIDE DERIVATIVES AS ANTIMICROBIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-23 WO disclosed