SCHEMBL14969093

SCHEMBL14969093

O=C(O)C1CC(Oc2ccc(-c3ccc(-c4nc5cc(F)ccc5[nH]4)c(F)c3)cn2)C1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.56
KCNH2 Q12809 8/20 0.56
ADORA2A P29274 3/20 0.48
SOAT1 P35610 3/20 0.47
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969139 1.00 DGAT1 (0.56) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14971565 1.00 DGAT1 (0.56) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14972173 0.93 DGAT1 (0.66) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL14972187 0.91 DGAT1 (0.59) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14969271 0.90 DGAT1 (0.52) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14971844 0.90 DGAT1 (0.52) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14969212 0.90 DGAT1 (0.52) DGAT1KCNH2ADORA2ASOAT1DHODH
SCHEMBL14972233 0.90 DGAT1 (0.45) DGAT1KCNH2ADORA2ADHODH
SCHEMBL14972175 0.88 DGAT1 (0.75) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL14972191 0.88 DGAT1 (0.75) DGAT1KCNH2ADORA2ASOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed