SCHEMBL14969288

SCHEMBL14969288

CCOC(=O)C1(C(=O)OCC)CC(Oc2ccc(Br)cn2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.49
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 5/20 0.37
MAPT P10636 3/20 0.37
CPB2 Q96IY4 1/20 0.37
HCRTR2 O43614 2/20 0.36
HSD11B1 P28845 2/20 0.36
HSD11B2 P80365 1/20 0.36
MAPK1 P28482 2/20 0.35
MEN1 O00255 1/20 0.35
S1PR4 O95977 1/20 0.35
LMNA P02545 1/20 0.35
S1PR1 P21453 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPC1 O15118 2/20 0.34
TP53 P04637 1/20 0.34
EPHX2 P34913 1/20 0.34
HCRTR1 O43613 2/20 0.34
MMP1 P03956 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971567 0.82 DGAT1 (0.57) DGAT1KDM4ERAB9AMAPTCPB2
SCHEMBL14971934 0.82 DGAT1 (0.57) DGAT1KDM4ERAB9AMAPTCPB2
SCHEMBL14968100 0.82 DGAT1 (0.57) DGAT1KDM4ERAB9AMAPTCPB2
SCHEMBL14968065 0.79 DGAT1 (0.50) DGAT1KDM4EMAPTHSD11B1MAPK1
SCHEMBL669097 0.79 DGAT1 (0.50) DGAT1KDM4EMAPTHSD11B1MAPK1
SCHEMBL14968084 0.79 DGAT1 (0.50) DGAT1KDM4EMAPTHSD11B1MAPK1
SCHEMBL14967794 0.77 DGAT1 (0.51) DGAT1KDM4ERAB9AMAPTHCRTR2
SCHEMBL14967861 0.77 DGAT1 (0.48) DGAT1KDM4EMAPTHCRTR2MAPK1
SCHEMBL22907265 0.76 DGAT1 (0.43) DGAT1KDM4ERAB9AMAPTHCRTR2
SCHEMBL29547742 0.76 DGAT1 (0.43) DGAT1KDM4ERAB9AMAPTHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed