SCHEMBL14971920

SCHEMBL14971920

O=C(O)[C@H]1C[C@@H](Oc2ncc(-c3ccc(-c4nc5c(F)cc(F)cc5[nH]4)c(F)c3)cn2)C1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 13/20 0.51
DGAT1 O75907 4/20 0.47
KCNH2 Q12809 3/20 0.47
SOAT1 P35610 1/20 0.47
PARP1 P09874 5/20 0.46
ADORA2A P29274 1/20 0.44
SSTR5 P35346 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971877 0.90 DGAT1 (0.56) DHODHDGAT1KCNH2SOAT1PARP1
SCHEMBL14972171 0.90 DGAT1 (0.56) DHODHDGAT1KCNH2SOAT1PARP1
SCHEMBL14971791 0.87 DHODH (0.45) DHODHDGAT1KCNH2SOAT1PARP1
SCHEMBL14972233 0.86 DGAT1 (0.45) DHODHDGAT1KCNH2PARP1ADORA2A
SCHEMBL14972249 0.84 DGAT1 (0.49) DHODHDGAT1KCNH2ADORA2A
SCHEMBL14969110 0.84 DGAT1 (0.49) DHODHDGAT1KCNH2ADORA2A
SCHEMBL14971597 0.84 DGAT1 (0.67) DHODHDGAT1KCNH2SOAT1PARP1
SCHEMBL14972256 0.83 DGAT1 (0.49) DHODHDGAT1KCNH2SOAT1ADORA2A
SCHEMBL14972239 0.83 DGAT1 (0.47) DHODHDGAT1KCNH2SOAT1ADORA2A
SCHEMBL14972255 0.82 DGAT1 (0.51) DHODHDGAT1KCNH2PARP1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed