SCHEMBL14972144

SCHEMBL14972144

Cc1ccc(OC(C)c2ccc(C(=O)NCc3c(C)cc(C)nc3O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.42
MMP13 P45452 4/20 0.42
MAPK14 Q16539 2/20 0.42
CYP3A4 P08684 2/20 0.42
MMP2 P08253 1/20 0.42
STAT3 P40763 1/20 0.42
HTT P42858 1/20 0.42
POLB P06746 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 3/20 0.40
TP53 P04637 3/20 0.39
CHRNA7 P36544 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969773 0.92 PPARA (0.45) SMN1; SMN2MAPK14CYP3A4POLBNPC1
SCHEMBL14969416 0.92 PPARA (0.45) SMN1; SMN2MAPK14CYP3A4POLBNPC1
SCHEMBL14966982 0.92 PPARA (0.45) SMN1; SMN2MAPK14CYP3A4POLBNPC1
SCHEMBL14967406 0.92 SMN1; SMN2 (0.45) SMN1; SMN2MAPK14POLBRAB9AALDH1A1
SCHEMBL14966658 0.92 SMN1; SMN2 (0.45) SMN1; SMN2MAPK14POLBRAB9AALDH1A1
SCHEMBL14967419 0.92 SMN1; SMN2 (0.45) SMN1; SMN2MAPK14POLBRAB9AALDH1A1
SCHEMBL14967264 0.91 SMN1; SMN2 (0.42) SMN1; SMN2MMP13MAPK14CYP3A4MMP2
SCHEMBL14966798 0.90 KLKB1 (0.44) SMN1; SMN2MMP13MAPK14HTTPOLB
SCHEMBL14967253 0.89 MEN1 (0.41) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL14966828 0.87 SMN1; SMN2 (0.41) SMN1; SMN2POLBNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9206128-B2 Modulators of methyl modifying enzymes, compositions and uses thereof CONSTELLATION PHARMACEUTICALS, INC. (US) 2015-12-08 US disclosed
US-9206128-B2 Modulators of methyl modifying enzymes, compositions and uses thereof CONSTELLATION PHARMACEUTICALS, INC. (US) 2015-12-08 US disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed